Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_01278
Ion Channel
Voltage-gated potassium channel subfamily D member 3
Peptide Function
Blocker
Gene Name
KCND3
Activity Data (nM)
IC50
9.6 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified
Sequence Information
Peptide Sequence
YCQKWMWTCDSKRACCEGLRCKLWCRKII
Peptide UniProt Accession
UniParc
UPI0001627736
Peptide Synonyms/Alias
JzTx-V; β/κ-Theraphotoxin-Cg2a; β/κ-TRTX-Cg2a; Peptide F8-15.73; Beta-theraphotoxin-Cj2a
Peptide Species
Chilobrachys guangxiensis (Chinese earth tiger tarantula) (Chilobrachys jingzhao)
Peptide Name
Beta/kappa-theraphotoxin-Cg2a
CAS Number
Not available
Experimental Conditions
pH
pH 7.2
Holding Potential (mV)
−80 mV
Temperature
25 °C
Test Method
Patch-clamping
Test Species
HEK293T cell (Homo sapiens embryonic kidney 293T cell)
Binding Information
Binding Site
Not specified
Binding Site Residue
Not specified
Ion Channel Information
Gene Abbreviation (ABB)
VGKCs
Ion Channel UniProt Accession
Source Organism
Homo sapiens (Human)
References & Disease Information
Disease
Not specified
PubChem CID
Not available
URL
Not available
PMID
Patent
Not available